| Generic Name | Brand Name | View All PK Information |
| Acarbose | Precose ® | |
| Acetohexamide | Dymelor ® | |
| Buformin | ® | |
| Chlorpropamide | ® | |
| Glibenclamide | ® | |
| Glibornuride | ® | |
| Gliclazide | ® | |
| Glimepiride | ® | |
| Glipizide | ® | |
| Gliquidone | ® | |
| Insulin | ® | |
| Metformin | ® | |
| Miglitol | ® | |
| Nateglinide | ® | |
| Orlistat | ® | |
| Phenformin | ® | |
| Raglitazar | ® | |
| Repaglinide | ® | |
| Rosiglitazone | ® | |
| Tolazamide | ® | |
| Tolbutamide | ® | |
| Tolrestat | ® | |
| Zopolrestat | ® |